Bioactive Small Molecules
![Medchemexpress LLC N-[[4-(benzamidocarbamoyl)cyclohexyl]methyl]-2-nitro-4-(trifluoromethyl)benzenesulfonamide | 263849-50-9 | 99.1% | 528.50 | C22H23F3N4O6S | 100 MG](https://assets.fishersci.com/TFS-Assets/CCG/product-images/5000241204.png-250.jpg)
Medchemexpress LLC N-[[4-(benzamidocarbamoyl)cyclohexyl]methyl]-2-nitro-4-(trifluoromethyl)benzenesulfonamide | 263849-50-9 | 99.1% | 528.50 | C22H23F3N4O6S | 100 MG
S 25585 is a potent, selective neuropeptide Y (NPY) Y5 receptor antagonist used as a research compound in preclinical studies of appetite regulation and NPY signaling. It is supplied as a high-purity solid with documented storage stability for laboratory use.
- High purity (99.1%).
- Molecular weight 528.50.
- Chemical formula C22H23F3N4O6S.
- Solid, white to off-white physical form.
- Documented storage stability at room temperature and in solvent at low temperatures.
- Intended for preclinical NPY receptor and appetite regulation research.
- Available in small-mass packages suitable for laboratory experiments.
Cayman Chemical OrnIpresInacetate 5mg
A vasopressin V1A receptor agonist; selectively induces reporter gene expression in HEK293 cells expressing vasopressin V1A and V2 receptors in reporter assays (EC50s = 0.69 and 0.45 nM, respectively, for the human receptors) over cells expressing vasopressin V1B receptors; selective for vasopressin V1A and V2 receptors over the vasopressin V1B receptor and oxytocin receptor (EC50s = 7.5 and 71 nM, respectively); increases arterial blood pressure in rats at 0.1 nmol/kg
Selleck Chemical LLC OSI-027 S2624-10mM/1mL
OSI-027 (ASP4786 CERC 006 AEVI-006) is a selective and potent dual inhibitor of mTORC1 and mTORC2 with IC50 of 22 nM and 65 nM in cell-free assays and more than 100-fold selectivity observed for mTOR than PI3K PI3K PI3K or DNA-PK OSI-027 induces autophagy in cancer cells
Cayman Chemical 6AmIno8trIfluoromethylphen 5mg
An antiprion agent; inhibits protein folding activity of the ribosome at 150 µM; directly competes with protein substrates for the ribosomal active site
Selleck Chemical LLC Securinine S9249-1MG
Securinine a major natural alkaloid product from the root of the plant Securinega suffruticosa acts as a -amino butyric acid (GABA) receptor antagonist
Selleck Chemical LLC Coixol S9253-5MG
Coixol (6-methoxybenzoxazolone MBOA) acts as a central muscle relaxant with an anti-convulsant effect
Medchemexpress LLC Decanoyl-RVKR-CMK | 150113-99-8 | MFCD00798792 | 98.0% | 744.41 | C34H66ClN11O5 | 10 MG
Decanoyl-RVKR-CMK is a peptidic inhibitor of subtilisin/Kex2p-like proprotein convertases, including furin. It blocks envelope glycoprotein precursor processing and gp160 maturation, and has been used to inhibit HIV-1 and HIV-2 replication in cell models. Typical applications include studies of viral glycoprotein processing, secretory pathway regulation, and protease biology.
- Inhibits furin and related proprotein convertases.
- Blocks envelope glycoprotein precursor processing and gp160 maturation.
- Used to probe viral replication and glycoprotein processing in cell models.
- Supplied as a purified research reagent (purity 98.0%).
- Molecular weight 744.41; formula C34H66ClN11O5.
Cayman Chemical ANTIBODY ACPT-I 10mg
An mGluR4a and mGluR8 agonist (EC50s = 7.2 and 8.2 µM, respectively); has no effect on mGluR1a or mGluR2; reduces cell death following oxygen-glucose deprivation in primary neuronal cultures using concentrations of 1-200 µM; reduces cell death in a rat model of middle cerebral artery occlusion when used at a dose of 30 mg/kg; reduces the incidence of clonic seizures in various seizure models in mice and rats (ED50s = 0.08-49.3 nM, i.c.v.); has anxiolytic-like effects in mice and rats that can be blocked by 5-HT1A and GABAA receptor antagonists